Program

42
5
1
1
1

Journal Year Published

7
2
5
3
7
4
6
1
3
3
1

Author

42
183
175
135
134
127
119
118
115
108
90
87
81
74
57
52
50
44
43
34

Category

26
12
11
10
2
1
1

Keyword

22
14
9
8
7
6
6
5
5
4
4
4
3
3
3
3
3
3
3
3

Journal

10
3
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1

NCATS Publications

Oxadiazole 2-oxides are toxic to the human hookworm, Ancylostoma ceylanicum, however glutathione reductase is not the primary target.


Treger RS, Cook AG, Rai Bantukallu G, Maloney DJ, Simeonov A, Jadhav A, Thomas C, Williams DL, Cappello M, Vermeire JJ


Int J Parasitol Drugs Drug Resist , (2), 171-177, 2012.

Article Pubmed

Sample image from publication page

Integration of pro-inflammatory cytokines, 12-lipoxygenase and NOX-1 in pancreatic islet beta cell dysfunction.


Weaver JR, Holman TR, Imai Y, Jadhav A, Kenyon V, Maloney DJ, Nadler JL, Rai Bantukallu G, Simeonov A, Taylor-Fishwick DA


Mol. Cell. Endocrinol. , (358), 88-95, 2012.

Article Pubmed

Sample image from publication page

Protein kinase C regulation of 12-lipoxygenase-mediated human platelet activation.


Yeung J, Apopa PL, Vesci J, Kenyon V, Rai Bantukallu G, Jadhav A, Simeonov A, Holman TR, Maloney DJ, Boutaud O, Holinstat M


Mol. Pharmacol. , (81), 420-30, 2012.

Article Pubmed

Sample image from publication page

Discovery of potent and selective inhibitors of human platelet-type 12- lipoxygenase.


Kenyon V, Rai Bantukallu G, Jadhav A, Schultz L, Armstrong M, Jameson JB, Perry S, Joshi N, Bougie JM, Leister W, Taylor-Fishwick DA, Nadler JL, Holinstat M, Simeonov A, Maloney DJ, Holman TR


J. Med. Chem. , (54), 5485-97, 2011.

Article Pubmed

Sample image from publication page

Quantitative high-throughput screening identifies 8-hydroxyquinolines as cell-active histone demethylase inhibitors.


King ON, Li XS, Sakurai M, Kawamura A, Rose NR, Ng SS, Quinn AM, Rai Bantukallu G, Mott BT, Beswick P, Klose RJ, Oppermann U, Jadhav A, Heightman TD, Maloney DJ, Schofield CJ, Simeonov A


PLoS ONE , (5), e15535, 2010.

Article Pubmed

Sample image from publication page

Discovery of potent and selective inhibitors of human reticulocyte 15-lipoxygenase-1.


Rai Bantukallu G, Kenyon V, Jadhav A, Schultz L, Armstrong M, Jameson JB, Hoobler E, Leister W, Simeonov A, Holman TR, Maloney DJ


J. Med. Chem. , (53), 7392-404, 2010.

Article Pubmed

Sample image from publication page

Molecular basis for the high-affinity binding and stabilization of firefly luciferase by PTC124.


Auld DS, Lovell S, Thorne N, Lea WA, Maloney DJ, Shen M, Rai Bantukallu G, Battaile KP, Thomas C, Simeonov A, Hanzlik RP, Inglese J


Proc. Natl. Acad. Sci. U.S.A. , (107), 4878-83, 2010.

Article Pubmed

Sample image from publication page

Structure mechanism insights and the role of nitric oxide donation guide the development of oxadiazole-2-oxides as therapeutic agents against schistosomiasis.


Rai Bantukallu G, Sayed AA, Lea WA, Luecke HF, Chakrapani H, Prast-Nielsen S, Jadhav A, Leister W, Shen M, Inglese J, Austin C, Keefer L, Arnér ES, Simeonov A, Maloney DJ, Williams DL, Thomas C


J. Med. Chem. , (52), 6474-83, 2009.

Article Pubmed

Sample image from publication page