Program

42
5
1
1
1

Journal Year Published

1
7
2
5
3
7
4
6
1
3
3
1

Author

43
201
181
149
139
133
133
125
123
108
105
95
82
78
63
62
54
50
46
43

Category

26
12
11
10
2
1
1

Keyword

22
14
9
8
7
6
6
5
5
4
4
4
3
3
3
3
3
3
3
3

Journal

10
3
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1

NCATS Publications

A furoxan-amodiaquine hybrid as a potential therapeutic for three parasitic diseases().


Mott BT, Cheng KC, Guha R, Kommer VP, Williams DL, Vermeire JJ, Cappello M, Maloney DJ, Rai Bantukallu G, Jadhav A, Simeonov A, Inglese J, Posner GH, Thomas C


Medchemcomm , (3), 1505-1511, 2012.

Article Pubmed

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Oxadiazole 2-oxides are toxic to the human hookworm, Ancylostoma ceylanicum, however glutathione reductase is not the primary target.


Treger RS, Cook AG, Rai Bantukallu G, Maloney DJ, Simeonov A, Jadhav A, Thomas C, Williams DL, Cappello M, Vermeire JJ


Int J Parasitol Drugs Drug Resist , (2), 171-177, 2012.

Article Pubmed

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Integration of pro-inflammatory cytokines, 12-lipoxygenase and NOX-1 in pancreatic islet beta cell dysfunction.


Weaver JR, Holman TR, Imai Y, Jadhav A, Kenyon V, Maloney DJ, Nadler JL, Rai Bantukallu G, Simeonov A, Taylor-Fishwick DA


Mol. Cell. Endocrinol. , (358), 88-95, 2012.

Article Pubmed

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Protein kinase C regulation of 12-lipoxygenase-mediated human platelet activation.


Yeung J, Apopa PL, Vesci J, Kenyon V, Rai Bantukallu G, Jadhav A, Simeonov A, Holman TR, Maloney DJ, Boutaud O, Holinstat M


Mol. Pharmacol. , (81), 420-30, 2012.

Article Pubmed

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Discovery of potent and selective inhibitors of human platelet-type 12- lipoxygenase.


Kenyon V, Rai Bantukallu G, Jadhav A, Schultz L, Armstrong M, Jameson JB, Perry S, Joshi N, Bougie JM, Leister W, Taylor-Fishwick DA, Nadler JL, Holinstat M, Simeonov A, Maloney DJ, Holman TR


J. Med. Chem. , (54), 5485-97, 2011.

Article Pubmed

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Quantitative high-throughput screening identifies 8-hydroxyquinolines as cell-active histone demethylase inhibitors.


King ON, Li XS, Sakurai M, Kawamura A, Rose NR, Ng SS, Quinn AM, Rai Bantukallu G, Mott BT, Beswick P, Klose RJ, Oppermann U, Jadhav A, Heightman TD, Maloney DJ, Schofield CJ, Simeonov A


PLoS ONE , (5), e15535, 2010.

Article Pubmed

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Discovery of potent and selective inhibitors of human reticulocyte 15-lipoxygenase-1.


Rai Bantukallu G, Kenyon V, Jadhav A, Schultz L, Armstrong M, Jameson JB, Hoobler E, Leister W, Simeonov A, Holman TR, Maloney DJ


J. Med. Chem. , (53), 7392-404, 2010.

Article Pubmed

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Molecular basis for the high-affinity binding and stabilization of firefly luciferase by PTC124.


Auld DS, Lovell S, Thorne N, Lea WA, Maloney DJ, Shen M, Rai Bantukallu G, Battaile KP, Thomas C, Simeonov A, Hanzlik RP, Inglese J


Proc. Natl. Acad. Sci. U.S.A. , (107), 4878-83, 2010.

Article Pubmed

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