Program

33
3
1

Journal Year Published

3
1
4
3
4
1
7
3
1
1
3
4
1
2

Author

38
201
181
149
139
133
133
125
123
108
105
95
82
78
63
62
54
50
46
43
43

Category

20
14
10
5
2
1
1
1

Keyword

14
7
6
6
6
6
5
5
5
4
4
4
3
3
3
3
3
3
3
2

Journal

6
3
3
2
2
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1

NCATS Publications

Synthesis and structure-activity relationship studies of 4-((2-hydroxy-3-methoxybenzyl)amino)benzenesulfonamide derivatives as potent and selective inhibitors of 12-lipoxygenase.


Luci D, Jameson JB, Yasgar A, Diaz G, Joshi N, Kantz A, Markham K, Perry S, Kuhn N, Yeung J, Kerns EH, Schultz L, Holinstat M, Nadler JL, Taylor-Fishwick DA, Jadhav A, Simeonov A, Holman TR, Maloney DJ


J. Med. Chem. , (57), 495-506, 2014.

Article Pubmed

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A fluorescence-based high throughput assay for the determination of small molecule-human serum albumin protein binding.


McCallum MM, Pawlak AJ, Shadrick WR, Simeonov A, Jadhav A, Yasgar A, Maloney DJ, Arnold LA


Anal Bioanal Chem , (406), 1867-75, 2014.

Article Pubmed

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Disrupting malaria parasite AMA1-RON2 interaction with a small molecule prevents erythrocyte invasion.


Srinivasan P, Yasgar A, Luci D, Beatty WL, Hu X, Andersen J, Narum DL, Moch JK, Sun H, Haynes JD, Maloney DJ, Jadhav A, Simeonov A, Miller LH


Nat Commun , (4), 2261, 2013.

Article Pubmed

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Peroxisome proliferation-activated receptor δ agonist GW0742 interacts weakly with multiple nuclear receptors, including the vitamin D receptor.


Nandhikonda P, Yasgar A, Baranowski AM, Sidhu PS, McCallum MM, Pawlak AJ, Teske K, Feleke B, Yuan NY, Kevin C, Bikle DD, Ayers SD, Webb P, Rai Bantukallu G, Simeonov A, Jadhav A, Maloney D, Arnold LA


Biochemistry , (52), 4193-203, 2013.

Article Pubmed

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High-throughput identification of promiscuous inhibitors from screening libraries with the use of a thiol-containing fluorescent probe.


McCallum MM, Nandhikonda P, Temmer JJ, Eyermann C, Simeonov A, Jadhav A, Yasgar A, Maloney D, Arnold AL


J Biomol Screen , (18), 705-13, 2013.

Article Pubmed

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Preparation of FRET reporters to support chemical probe development.


Foley TL, Yasgar A, Garcia CJ, Jadhav A, Simeonov A, Burkart MD


Org. Biomol. Chem. , (8), 4601-6, 2010.

Article Pubmed

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